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Journal Article 2

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2023 1

2009 1

Keywords

(R)-(+)-1(1-naphthyl)ethylamine 1

Amine transaminase 1

Co-evolution 1

Trade-off 1

antimicrobial 1

microwave-assisted synthesis 1

naphthyl 1

thiazolidin-4-one 1

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Microwave-assisted synthesis and antimicrobial activities of 2-aryl-3-(naphthalene-1 or 2-yl)-1,3-thiazolidin-4-ones

Hua CHEN, Yanan LI, Jie BAI, Lian ZHAO, Xiangguo YUAN, Xiaoliu LI, Keqiang CAO

Frontiers of Chemical Science and Engineering 2009, Volume 3, Issue 2,   Pages 186-191 doi: 10.1007/s11705-009-0004-0

Abstract: 2-aryl-3-(naphthalene-1 or 2-yl)-1,3-thiazolidin-4-ones and were synthesized in 41%-67% yield by using microwave-assisted one-pot protocol. The structures of the new compounds , , , , , , and - were confirmed by IR, NMR, MS, and elemental analysis. The antimicrobial activities of the compounds against pv. lachrymans (Smith et Bryan) Young, Dye & Wilkie, Pers., and Blum. were examined. Some of the compounds showed good antifungical activity against Blum.

Keywords： microwave-assisted synthesis     naphthyl     thiazolidin-4-one     antimicrobial    

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Pocket Modification of ω-Amine Transaminase AtATA for Overcoming the Trade-Off between Activity and Stability Toward 1-Acetonaphthone Article

Jiaren Cao, Fangfang Fan, Changjiang Lyu, Sheng Hu, Weirui Zhao, Jiaqi Mei, Shuai Qiu, Lehe Mei, Jun Huang

Engineering 2023, Volume 30, Issue 11,   Pages 203-214 doi: 10.1016/j.eng.2023.04.009

Abstract: aliquot of 1-acetonaphthone in a 50 mL scaledup system to the desired product, (R)-(+)-1(1-naphthyl

Keywords： Trade-off     Co-evolution     Amine transaminase     (R)-(+)-1(1-naphthyl)ethylamine    

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Microwave-assisted synthesis and antimicrobial activities of 2-aryl-3-(naphthalene-1 or 2-yl)-1,3-thiazolidin-4-ones

Hua CHEN, Yanan LI, Jie BAI, Lian ZHAO, Xiangguo YUAN, Xiaoliu LI, Keqiang CAO

Journal Article

Pocket Modification of ω-Amine Transaminase AtATA for Overcoming the Trade-Off between Activity and Stability Toward 1-Acetonaphthone

Jiaren Cao, Fangfang Fan, Changjiang Lyu, Sheng Hu, Weirui Zhao, Jiaqi Mei, Shuai Qiu, Lehe Mei, Jun Huang

Journal Article